司美替尼
司美替尼
MEK1/2抑制剂;司美替尼
Selumetinib
MEK1/2抑制剂;司美替尼
Selumetinib
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产品编号: CSR254000
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CAS号: 606143-52-6
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分子式:C17H15BrClFN4O3
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分子量:457.68
英文别名:
ARRY 142886;AZD 6244
参考文献:
Ciardiello, F., et al.: Clin. Cancer Res., 7, 1459 (2001), Hidalgo, M., et al.: J. Clin. Oncol., 19, 3267 (2001),
It is a tight-binding, uncompetitive inhibitor of mitogen-activated protein kinase kinases (MEK) 1 and 2 currently in clinical development.
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