Pictrelisib
Pictrelisib
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Pictrelisib
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Pictrelisib
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产品编号: CGR601510
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CAS号: 957054-30-7
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分子式:C23H27N7O3S2
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分子量:513.64
英文别名:
GDC-0941;Pictilisib
SMILES:
C(OC([2H])([2H])C([2H])(C([2H])([2H])OC(=O)CCCCCCCCCCCCCCC)O)(=O)CCCCCCCCCCCCCCC
参考文献:
Jeffrey J.W., et al.: Clinical. Cancer. Rsch., 10, 1078 (2012); Murray, J.M., et al.: J. Medn. Chem., 55, 7686 (2012);
GDC-0941 is a potent and selective oral inhibitor of the class I PI3K. GDC-0941 demonstrated broad spectrum of activity in breast, ovarian, lung, and prostate cancer models. Studies has also shown GDC-0941 may enhance anti-tumor activity of Docetaxel (D49
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