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依维莫司
雷帕霉素衍生物;依维莫司;42-O-(2-羟基)乙基雷帕霉素
Everolimus
  • 产品编号: CER945400

  • CAS号: 159351-69-6

  • 分子式:C53H83NO14

  • 分子量:958.22

英文别名:
40-O-(2-Hydroxyethyl)rapamycin; 42-O-(2-Hydroxy)ethyl Rapamycin; Afinitor; Certican; RAD; RAD 001; SDZ-RAD; XIENCE V
熔点:
110-115°C
可溶性:
Chloroform, Methanol
性状:
Off White to Pale Yellow Solid
储存条件:
Hygroscopic, Store under Inert atmosphere -20°C Freezer
参考文献:
Dumont, F.J., et al.: Curr. Opin. Invest. Drugs, 2, 1220 (2001), Kovarik, J. M., et al.: Clin. Pharmacol. Ther., 69, 48 (2001), Nashan, B., et al.: Ther. Drug Monit., 24, 53 (2002),
Everolimus Macrolide immunosuppressant; Everolimus is a derivative of Rapamycin. Everolimus inhibits cytokine-mediated lymphocyte proliferation.
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