依克立达-d4
依克立达-d4
依克立达-d4;依拉克达-d4 (混合物)
Elacridar-d4
依克立达-d4;依拉克达-d4 (混合物)
Elacridar-d4
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产品编号: CER489002
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CAS号: 1189481-51-3
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分子式:C34H29D4N3O5
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分子量:567.67
英文别名:
N-[4-[2-(3,4-Dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)ethyl-d4]phenyl]-9,10-dihydro-5-methoxy-9-oxo-4-acridinecarboxamide; GF 120918-d4;
GG 918-d4; GW 0918-d4;
熔点:
198-200°C
可溶性:
DMSO, Methanol
性状:
Yellow Solid
储存条件:
-20˚C Freezer
参考文献:
Neville, K., et al.: Clin. Cancer Res., 10, 2525 (2004), Reardon, D., et al.: J. Clin. Oncol. 23, 9359 (2005), Pan, G., et al.: Drug Metab. Dispos., 35, 1165 (2007).
A prototypical BCRP inhibitor. Inhibits the Bcrp1-mediated transport.
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