皮啡肽三氟乙酸盐
皮啡肽三氟乙酸盐
Dermorphin Trifluoroacetate
皮啡肽三氟乙酸盐
Dermorphin Trifluoroacetate
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产品编号： CDR281940
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CAS号： 78331-26-7
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分子式：C43H51F3N8O12
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分子量：916.9
英文别名：
L-Tyrosyl-D-alanyl-L-phenylalanylglycyl-L-tyrosyl-L-prolyl-L-serinamide Trifluoroacetate; Tyr-D-Ala-Phe-Gly-Tyr-Pro-Ser-NH2 TFA Salt;
熔点：
157-162°C
可溶性：
DMSO, Methanol
性状：
白色固体
SMILES：
O=C([O-])C1C(=CC=CC=1)C(O)C2C(CC(N3C(=O)NC(=O)C(I)=C3)O2)(O)C4C(=CC=CC=4)C(=O)[O-]
储存条件：
-20°C
参考文献：
Erspamer, V. et al.: Proc. Nat. Acad. Sci. U.S.A., 86, 5188 (1989); Negri, L. et al.: Hand. Biol. Act. Pep., 268 (2006); Broccardo, M. et al.: Br. J. Pharmacol., 73, 625 (1981);
Dermorphin is a hepta-peptide and a natural opioid initially isolated from the skin of South American hylid frogs Phyllomedusinae. Dermorphin binds as an agonist with high potency and selectivity to mu-opioid receptors. Dermorphin is about 30-40 times more potent than Morphine.
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